/DISCLAIMER · RESEARCH_COMPOUND

This page is reference information only. Most compounds described here are research chemicals, not FDA-approved medications. MyTRT does not sell, recommend, or endorse the use of these substances. Always consult a qualified physician.

/5_AMINO_1MQ
Small Molecule

5-Amino-1MQ

Nicotinamide N-methyltransferase Inhibitor

/HALF_LIFE
Not well characterized
/DELIVERY
Oral

/WHAT_IT_IS

5-Amino-1MQ is a potent and selective small-molecule inhibitor of nicotinamide N-methyltransferase (NNMT), an enzyme that methylates nicotinamide to 1-methylnicotinamide, thereby modulating NAD⁺ metabolism and influencing energy expenditure and adiposity.

/USAGE

Used in research to study NNMT activity, NAD⁺ salvage pathways, obesity, type 2 diabetes, and metabolic regulation.

/MECHANISM_OF_ACTION

Binds to the active site of NNMT, preventing methylation of nicotinamide, which leads to increased intracellular NAD⁺ levels, enhanced mitochondrial function, and reduced lipogenesis.

Reported Benefits

  • +Increased NAD⁺ levels
  • +Enhanced mitochondrial function
  • +Reduced adiposity in diet-induced obesity models
  • +Improved glucose tolerance

Reported Side Effects

  • Not well characterized in humans
  • Potential off-target effects at high doses

/RESEARCH_NOTES

In mouse studies, 5-Amino-1MQ reverses diet-induced obesity without affecting food intake and shows high selectivity over other methyltransferases. Human data are limited.

/REFERENCE

https://pubmed.ncbi.nlm.nih.gov/35013352/
/TRACK_THIS

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Last reviewed: 2026-06-04 · Reference only. Not medical advice. Consult a qualified physician.