/DISCLAIMER · RESEARCH_COMPOUND

This page is reference information only. Most compounds described here are research chemicals, not FDA-approved medications. MyTRT does not sell, recommend, or endorse the use of these substances. Always consult a qualified physician.

/ARIMIDEX
Antiestrogen / Ancillary

Arimidex (Anastrozole)

Aromatase Inhibitor (AI)

/HALF_LIFE
Approximately 40–50 hours
/DELIVERY
Oral tablet or capsule

/WHAT_IT_IS

Arimidex (anastrozole) is a non-steroidal aromatase inhibitor that blocks the conversion of androgens into estrogen, reducing estrogen levels in the body.

/USAGE

Used clinically to treat hormone receptor‑positive breast cancer in postmenopausal women; off-label in men and bodybuilders for estrogen management, gynecomastia prevention, and testosterone therapy.

/MECHANISM_OF_ACTION

Reversibly inhibits aromatase enzyme, preventing the aromatization of testosterone and androstenedione into estradiol and estrone.

Reported Benefits

  • +Reduces estrogen levels
  • +Helps prevent gynecomastia
  • +Supports hormonal balance during TRT or steroid cycles
  • +Used in breast cancer treatment and prevention

Reported Side Effects

  • Hot flashes
  • Joint/muscle pain and stiffness
  • Fatigue or weakness
  • Bone mineral density reduction (osteopenia/osteoporosis)
  • Nausea
  • Rare allergic reactions or liver enzyme changes

/STACKED_WITH

Selective Estrogen Receptor Modulators (SERMs) like Tamoxifen or ClomidTestosterone (TRT)AIs like Letrozole for fine-tuning estrogen suppression

/RESEARCH_NOTES

Therapeutic dose of 1 mg/day yields ~97% aromatase inhibition; hepatic metabolism accounts for ~85% of elimination, excreted primarily via urine and feces. Noted off-label use in men for estrogen control :contentReference[oaicite:1]{index=1}.

/TRACK_THIS

Browse all 89 in the app.

MyTRT's in-app library has the same 89 peptide entries plus dosing notes, stack builders, and the ability to log them alongside your TRT protocol.

Last reviewed: 2026-06-04 · Reference only. Not medical advice. Consult a qualified physician.